Heln hpr (heralpha dbd) cell line

HELN were generated by transfection of cervical cancer HeLa cells with the ERE-betaGlobin-Luciferase-SV40-Neomycin plasmid.
HELN hPR cells were generated by transfection of HELN cells with the pSG5-puro plasmid pSG5-human PR (ER alpha DBD)-puromycin.
The plasmid ERE-betaGlob-Luc-SVNeo contains a luciferase gene driven by estrogen receptor responsive element (ERE) in front of beta-globin promoter and a neomycin phosphotransferase gene under the control of SV40 promoter.
The pSG5-puro plasmid pSG5-human PR (ER alpha DBD)-puromycin enables to express the human progesterone receptor in which the DNA binding domain (DBD) has been replaced by the estrogen receptor alpha DBD.

Interest / Relevance: These cells enable to measure the hPR estrogenic activity of environmental (water, sediments), human (blood, urine adipose tissue) or food (water, vegetables, meat) samples.

R5020 EC50 0.33 nM
Scientist's name: Patrick BALAGUER
Publications:
Garoche C, Ait-Aissa S, Boulahtouf Abdelhay, Creusot N, Bourguet W, Balaguer P, Brion F. Human and zebrafish nuclear progesterone receptors are differently activated by progestins. Environmental Science & Technology 2020 , 54 : 9510-18. Neale P, Grimaldi M, Boulahtouf A, Leusch F*, Balaguer P. Assessing species-specific differences for nuclear receptor activation for environmental water extracts. Water Research 2020, 185 : 116247. Kroupova HK, Grimaldi M, Sauer P, Borik A, Zalohova K, Balaguer P. Environmental water extracts differentially activate the zebrafish and human nuclear progesterone receptor. STOTEN. 2022 Nov 16:160232.

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